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1

Practical Synthesis of a 6-Triazolylazabicyclo[3.1.0]hexane

Sirois, Lauren E., Xu, Jie, Angelaud, Remy, Lao, David, Gosselin, Francis

Journal:

Organic Process Research & Development

Year:

2018

Language:

english

File:

PDF, 1.25 MB

english, 2018

2

Development of a Second-Generation, Highly Efficient Manufacturing Route for the HIV Integrase Inhibitor Raltegravir Potassium

Humphrey, Guy R., Pye, Philip J., Zhong, Yong-Li, Angelaud, Remy, Askin, David, Belyk, Kevin M., Maligres, Peter E., Mancheno, Danny E., Miller, Ross A., Reamer, Robert A., Weissman, Steven A.

Journal:

Organic Process Research & Development

Year:

2011

Language:

english

File:

PDF, 1.22 MB

english, 2011

3

Preparative Scale Synthesis of the Biaryl Core of Anacetrapib via a Ruthenium-Catalyzed Direct Arylation Reaction: Unexpected Effect of Solvent Impurity on the Arylation Reaction †

Ouellet, Stéphane G., Roy, Amélie, Molinaro, Carmela, Angelaud, Rémy, Marcoux, Jean-François, O’Shea, Paul D., Davies, Ian W.

Journal:

Journal of Organic Chemistry

Year:

2011

Language:

english

File:

PDF, 798 KB

english, 2011

4

Manufacturing Development and Genotoxic Impurity Control Strategy of the Hedgehog Pathway Inhibitor Vismodegib

Angelaud, Remy, Reynolds, Mark, Venkatramani, Cadapakam J., Savage, Scott, Trafelet, Huldreich, Landmesser, Thomas, Demel, Peter, Levis, Michael, Ruha, Olivier, Rueckert, Baerbel, Jaeggi, Heinz

Journal:

Organic Process Research & Development

Year:

2016

Language:

english

File:

PDF, 735 KB

english, 2016

5

A Practical Synthesis of α-Aryl Methyl Ketones via a Transition-Metal-Free Meerwein Arylation

Molinaro, Carmela, Mowat, Jeffrey, Gosselin, Francis, O'Shea, Paul D., Marcoux, Jean-François, Angelaud, Rémy, Davies, Ian W.

Journal:

Journal of Organic Chemistry

Year:

2007

Language:

english

File:

PDF, 135 KB

english, 2007

6

Process Development Overcomes a Challenging Pd-Catalyzed CâN Coupling for the Synthesis of RORc Inhibitor GDC-0022

Sirois, Lauren E., Lao, David, Xu, Jie, Angelaud, RÃ©my, Tso, Jerry, Scott, Brandon, Chakravarty, Paroma, Malhotra, Sushant, Gosselin, Francis

Journal:

Organic Process Research & Development

Year:

2020

Language:

english

File:

PDF, 1.55 MB

english, 2020

7

Optical rotation per refractive index unit, or enantiomeric (e) factor, for screening enantioselective catalysts through asymmetric activation or carbohydrates

Remy Angelaud, Yousuke Matsumoto, Toshinobu Korenaga, Kenichi Kudo, Masaaki Senda, Koichi Mikami

Journal:

Year:

2000

Language:

english

File:

PDF, 121 KB

english, 2000

8

Asymmetrische Aktivierung

Koichi Mikami, Masahiro Terada, Toshinobu Korenaga, Yousuke Matsumoto, Makoto Ueki, Rémy Angelaud

Journal:

Angewandte Chemie

Year:

2000

Language:

german

File:

PDF, 824 KB

german, 2000

9

Asymmetric Activation of Chiral Alkoxyzinc Catalysts by Chiral Nitrogen Activators for Dialkylzinc Addition to Aldehydes: Super High-Throughput Screening of Combinatorial Libraries of Chiral Ligands and Activators by HPLC-CD/UV and HPLC-OR/RIU Systems

Koichi Mikami, Rémy Angelaud, Kuiling Ding, Akihiro Ishii, Akito Tanaka, Naotaka Sawada, Kenichi Kudo, Masaaki Senda

Journal:

Chemistry - A European Journal

Year:

2001

Language:

english

File:

PDF, 226 KB

english, 2001

10

Asymmetric Activation

Koichi Mikami, Masahiro Terada, Toshinobu Korenaga, Yousuke Matsumoto, Makoto Ueki, Rémy Angelaud

Journal:

Angewandte Chemie International Edition

Year:

2000

Language:

english

File:

PDF, 724 KB

english, 2000

11

ChemInform Abstract: Radical Deuteration of α-Selenylated-β-silylsulfoxides.

R. ANGELAUD, Y. LANDAIS

Journal:

Year:

1997

File:

PDF, 31 KB

1997

12

ChemInform Abstract: Asymmetric Amino-Hydroxylation of Dienylsilanes. An Efficient Route to Aminocyclitols.

R. ANGELAUD, Y. LANDAIS, K. SCHENK

Journal:

Year:

1997

File:

PDF, 30 KB

1997

13

ChemInform Abstract: Synthesis of Pseudo-Sugars Based on Desymmetrization of Dienylsilanes.

R. ANGELAUD, Y. LANDAIS

Journal:

Year:

1998

File:

PDF, 36 KB

1998

14

ChemInform Abstract: Stereocontrolled Access to Carba-C-disaccharides via Functionalized Dienylsilanes.

R. ANGELAUD, Y. LANDAIS, L. PARRA-RAPADO

Journal:

Year:

1998

File:

PDF, 30 KB

1998

15

ChemInform Abstract: Desymmetrization of Cyclohexadienylsilanes. Regio-, Diastereo-, and Enantioselective Access to Sugar Mimics.

Remy Angelaud, Odile Babot, Trevor Charvat, Yannick Landais

Journal:

Year:

2000

File:

PDF, 38 KB

2000

16

ChemInform Abstract: The Phenylthiocyclopropylsilyl Group: A Useful Latent Hydroxy Group.

Remy Angelaud, Yannick Landais

Journal:

Year:

2000

File:

PDF, 32 KB

2000

17

ChemInform Abstract: Asymmetric Activation

Koichi Mikami, Masahiro Terada, Toshinobu Korenaga, Yousuke Matsumoto, Makoto Ueki, Remy Angelaud

Journal:

Year:

2001

File:

PDF, 23 KB

2001

18

ChemInform Abstract: Asymmetric Activation of Chiral Alkoxyzinc Catalysts by Chiral Nitrogen Activators for Dialkylzinc Addition to Aldehydes: Super High-Throughput Screening of Combinatorial Libraries of Chiral Ligands and Activators by HPLC-CD/UV and HPLC-OR/RIU Systems.

Koichi Mikami, Remy Angelaud, Kuiling Ding, Akihiro Ishii, Akito Tanaka, Naotaka Sawada, Kenichi Kudo, Masaaki Senda

Journal:

Year:

2002

File:

PDF, 26 KB

2002

19

Desymmetrization of Cyclopentadienylsilane by Asymmetric Cyclopropanation.

Florent Allais, Remy Angelaud, Boris Camuzat-Dedenis, Karine Julienne, Yannick Landais

Journal:

Year:

2003

File:

PDF, 100 KB

2003

20

ChemInform Abstract: Regioselective SNAr Reactions of Substituted Difluorobenzene Derivatives: Practical Synthesis of Fluoroaryl Ethers and Substituted Resorcinols.

Stephane G. Ouellet, Anna Bernardi, Remy Angelaud, Paul D. O'Shea

Journal:

Year:

2009

File:

PDF, 30 KB

2009

21

Desymmetrisation of Cyclopentadienylsilane by Asymmetric Cyclopropanation

Florent Allais, Rémy Angelaud, Boris Camuzat-Dedenis, Karine Julienne, Yannick Landais

Journal:

European Journal of Organic Chemistry

Year:

2003

Language:

english

File:

PDF, 119 KB

english, 2003

22

The dimethyl(1-phenylthio)cyclopropylsilyl group as a masked hydroxyl group

Rémy Angelaud, Yannick Landais, Christian Maignan

Journal:

Tetrahedron Letters

Year:

1995

Language:

english

File:

PDF, 249 KB

english, 1995

23

Serendipitous discovery of a pH-dependant atropisomer bond rotation: Toward a write-protectable chiral molecular switch?

Christopher J. Welch, Mirlinda Biba, Philip Pye, Remy Angelaud, Melissa Egbertson

Journal:

Journal of Chromatography B

Year:

2008

Language:

english

File:

PDF, 389 KB

english, 2008

24

Radical deuteration of α-selenylated-β-silylsulfoxides

Rémy Angelaud, Yannick Landais

Journal:

Tetrahedron Letters

Year:

1997

Language:

english

File:

PDF, 265 KB

english, 1997

25

Asymmetric amino-hydroxylation of dienylsilanes. An efficient route to amino-cyclitols

Rémy Angelaud, Yannick Landais, Kurt Schenk

Journal:

Tetrahedron Letters

Year:

1997

Language:

english

File:

PDF, 246 KB

english, 1997

26

Stereocontrolled access to Carba-C-disaccharides via functionalized dienylsilanes

Rémy Angelaud, Yannick Landais, Liliana Parra-Rapado

Journal:

Tetrahedron Letters

Year:

1997

Language:

english

File:

PDF, 250 KB

english, 1997

27

Practical reduction of oxazolines to alcohols

Anna Bernardi, Stéphane G. Ouellet, Remy Angelaud, Paul D. O’Shea

Journal:

Tetrahedron Letters

Year:

2008

Language:

english

File:

PDF, 154 KB

english, 2008

28

Regioselective SNAr reactions of substituted difluorobenzene derivatives: practical synthesis of fluoroaryl ethers and substituted resorcinols

Stéphane G. Ouellet, Anna Bernardi, Remy Angelaud, Paul D. O’Shea

Journal:

Tetrahedron Letters

Year:

2009

Language:

english

File:

PDF, 1.60 MB

english, 2009

29

The Phenylthiocyclopropylsilyl Group: a Useful Latent Hydroxy Group

Rémy Angelaud, Yannick Landais

Journal:

Year:

2000

Language:

english

File:

PDF, 301 KB

english, 2000

30

Synthesis of pseudo-sugars based on desymmetrization of dienylsilanes

Rémy Angelaud, Yannick Landais

Journal:

Tetrahedron Letters

Year:

1997

Language:

english

File:

PDF, 261 KB

english, 1997

31

A Practical Synthesis of Renin Inhibitor MK-1597 (ACT-178882) via Catalytic Enantioselective Hydrogenation and Epimerization of Piperidine Intermediate

Molinaro, Carmela, Shultz, Scott, Roy, Amélie, Lau, Stephen, Trinh, Thao, Angelaud, Rémy, O’Shea, Paul D., Abele, Stefan, Cameron, Mark, Corley, Ed

Journal:

Journal of Organic Chemistry

Year:

2011

Language:

english

File:

PDF, 1.11 MB

english, 2011

32

Remote Electronic Control in the Regioselective Reduction of Succinimides: A Practical, Scalable Synthesis of EP4 Antagonist MF-310

Molinaro, Carmela, Gauvreau, Danny, Hughes, Gregory, Lau, Stephen, Lauzon, Sophie, Angelaud, Rémy, O’Shea, Paul D., Janey, Jacob, Palucki, Michael, Hoerrner, Scott R.

Journal:

Journal of Organic Chemistry

Year:

2009

Language:

english

File:

PDF, 783 KB

english, 2009

33

ChemInform Abstract: The Dimethyl(1-phenylthio)cyclopropylsilyl Group as a Masked Hydroxyl Group.

R. ANGELAUD, Y. LANDAIS, C. MAIGNAN

Journal:

Year:

1995

File:

PDF, 34 KB

1995

34

ChemInform Abstract: α-Silylthioethers as Masked Hydroxyl Groups

R. ANGELAUD, Y. LANDAIS, C. MAIGNAN

Journal:

Year:

1996

File:

PDF, 27 KB

1996

35

ChemInform Abstract: Desymmetrization of a Silyl-2,5-cyclohexadiene. Synthesis of (+)- Conduritol E and (-)-2-Deoxy-allo-inositol.

R. ANGELAUD, Y. LANDAIS

Journal:

Year:

1996

File:

PDF, 31 KB

1996

36

Desymmetrization of Cyclohexadienylsilanes. Regio-, Diastereo-, and Enantioselective Access to Sugar Mimics

Angelaud, Rémy, Babot, Odile, Charvat, Trevor, Landais, Yannick

Journal:

Journal of Organic Chemistry

Year:

1999

Language:

english

File:

PDF, 450 KB

english, 1999

37

Development of a Scalable Strategy for the Synthesis of PI3Kδ Inhibitors: Selective and Efficient Functionalization of Purine Derivatives

Carrera, Diane E., Sheng, PeiJue, Safina, Brian S., Li, Jun, Angelaud, Remy

Journal:

Organic Process Research & Development

Year:

2013

Language:

english

File:

PDF, 435 KB

english, 2013

38

Synthesis and evaluation of a broad range of chiral sulfides for asymmetric sulfur ylide epoxidation of aldehydes

Aggarwal, Varinder K., Angelaud, RÃ©my, Bihan, Dominique, Blackburn, Paul, Fieldhouse, Robin, Fonquerna, Silvia J., Ford, Gair D., Hynd, George, Jones, Elfyn, Jones, Ray V. H., Jubault, Philippe, Palm

Journal:

Journal of the Chemical Society Perkin Transactions 1

Year:

2001

Language:

english

File:

PDF, 360 KB

english, 2001

39

A Practical Synthesis of Renin Inhibitor MK-1597 (ACT-178882) via Catalytic Enantioselective Hydrogenation and Epimerization of Piperidine Intermediate

Molinaro, Carmela, Shultz, Scott, Roy, Amelie, Lau, Stephen, Trinh, Thao, Angelaud, Remy, O’Shea, Paul D., Abele, Stefan, Cameron, Mark, Corley, Ed, Funel, Jacques-Alexis, Steinhuebel, Dietrich, Weise

Journal:

Journal of Organic Chemistry

Year:

2012

Language:

english

File:

PDF, 154 KB

english, 2012

40

Synthesis of a β-Amino Acid Pharmacophore via a β-Lactam Intermediate

Angelaud, Rémy, Zhong, Yong-Li, Maligres, Peter, Lee, Jaemoon, Askin, David

Journal:

Journal of Organic Chemistry

Year:

2005

Language:

english

File:

PDF, 107 KB

english, 2005

41

Desymmetrization of a Silyl-2,5-cyclohexadiene. Synthesis of (+)-Conduritol E and (−)-2-Deoxy- allo -inositol

Angelaud, Rémy, Landais, Yannick

Journal:

Journal of Organic Chemistry

Year:

1996

Language:

english

File:

PDF, 117 KB

english, 1996

42

Development of an Expedient Process for the Multi-Kilogram Synthesis of Chk1 Inhibitor GDC-0425

Stumpf, Andreas, Cheng, Zhigang Ken, Wong, Brian, Reynolds, Mark, Angelaud, Remy, Girotti, James, Deese, Alan, Gu, Christine, Gazzard, Lewis

Journal:

Organic Process Research & Development

Year:

2015

Language:

english

File:

PDF, 766 KB

english, 2015

43

A Strecker approach to 2-substituted ethyl 5-aminothiazole-4-carboxylates

Cheng, Ken, McClory, Andrew, Walker, Whitney, Xu, Jie, Zhang, Haiming, Angelaud, Remy, Gosselin, Francis

Journal:

Tetrahedron Letters

Year:

2015

Language:

english

File:

PDF, 534 KB

english, 2015

44

Process Development of the Synthesis and Purification of a Reactive Immuno-PET Conjugate Intermediate

Carrera, Dr. Diane E., Nguyen, Tina, Medley, Colin D., Li, Yi, Angelaud, Remy, Gosselin, Francis

Journal:

Organic Process Research & Development

Year:

2016

Language:

english

File:

PDF, 542 KB

english, 2016

45

Development of an Efficient, Safe, and Environmentally Friendly Process for the Manufacture of GDC-0084

Stumpf, Andreas, McClory, Andrew, Yajima, Herbert, Segraves, Nathaniel, Angelaud, Remy, Gosselin, Francis

Journal:

Organic Process Research & Development

Year:

2016

Language:

english

File:

PDF, 990 KB

english, 2016

46

Magnesium Ethoxide Promoted Conversion of Nitriles to Amidines and Its Application in 5,6-Dihydroimidazobenzoxazepine Synthesis

Dalziel, Michael E., Deichert, Julie A., Carrera, Diane E., Beaudry, Danial, Han, Chong, Zhang, Haiming, Angelaud, Remy

Journal:

Organic Letters

Year:

2018

Language:

english

File:

PDF, 799 KB

english, 2018

47

ChemInform Abstract: A Strecker Approach to 2-Substituted Ethyl 5-Aminothiazole-4-carboxylates.

Cheng, Ken, McClory, Andrew, Walker, Whitney, Xu, Jie, Zhang, Haiming, Angelaud, Remy, Gosselin, Francis

Journal:

Year:

2016

File:

PDF, 20 KB

2016

48

Development of an Efficient Manufacturing Process for Reversible BTK Inhibitor GDC-0853

Zhang, Haiming, Cravillion, Theresa, Lim, Ngiap-Kie, Tian, Qingping, Beaudry, Danial, Defreese, Jessica, Fettes, Alec, James, Philippe, Linder, David, Malhotra, Sushant, Han, Chong, Angelaud, Remy, Go

Journal:

Organic Process Research & Development

Year:

2018

Language:

english

File:

PDF, 728 KB

english, 2018

49

A Telescoped Knochel-Hauser / Kumada-Corriu Coupling Strategy to Functionalized Aromatic Heterocycles

Clagg, Kyle, Hold, Sara, Kumar, Archana, Koenig, Stefan G., Angelaud, Remy

Journal:

Tetrahedron Letters

Year:

2018

Language:

english

File:

PDF, 672 KB

english, 2018

50

Study of a Competing Hydrodefluorination Reaction During the Directed ortho -Lithiation/Borylation of 2-Fluorobenzaldehyde

St-Jean, Frédéric, Piechowicz, Katarzyna A., Sirois, Lauren E., Angelaud, Rémy, Gosselin, Francis

Journal:

Organometallics

Year:

2018

Language:

english

File:

PDF, 1.56 MB

english, 2018